Eplivanserin hemifumarate is a potent and selective antagonist of the 5-HT2A receptor, exhibiting an IC50 of 5.8 nM in rat cortical membranes and a Kd of 1.14 nM. It demonstrates greater than 20-fold selectivity for the 5-HT2A subtype over 5-HT2B and 5-HT2C receptors. This compound is valuable for research focused on neuropharmacology and the modulation of serotonergic pathways in various biological processes.
Eplivanserin hemifumarate is a potent and selective antagonist of the 5-HT2A receptor, exhibiting an IC50 of 5.8 nM in rat cortical membranes and a Kd of 1.14 nM. It demonstrates greater than 20-fold selectivity for the 5-HT2A subtype over 5-HT2B and 5-HT2C receptors. This compound is valuable for research focused on neuropharmacology and the modulation of serotonergic pathways in various biological processes.
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