Eplivanserin is a potent, selective and orally available 5-HT2 receptor antagonist, with an IC50 of 5.8 nM in rat cortical membrane, and a Kd of 1.14 nM.
Eplivanserin is a potent, selective and orally available 5-HT2 receptor antagonist, with an IC50 of 5.8 nM in rat cortical membrane, and a Kd of 1.14 nM.
Targets
Target
Value
Product Information
Catalog Num
A21967
Formula
C19H21FN2O2
Molecular Weight
328.38
CAS Number
130579-75-8
SMILES
FC1=CC=CC=C1C(/C=C/C2=CC=C(O)C=C2)=N\OCCN(C)C
Synonyms
SR-46349, SR 46349, SR46349
Storage
Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula: