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Biological Activity
Eptapirone is a potent, selective, high efficacy 5-HT1A receptor agonist with marked anxiolytic and antidepressant potential. The affinity of F 11440 for 5-HT1A binding sites (pKi, 8.33) was higher than that of buspirone (pKi, 7.50), and somewhat lower than that of flesinoxan (pKi, 8.91). In vivo, F 11440 was 4- to 20-fold more potent than flesinoxan, and 30- to 60-fold more potent than buspirone.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 28.95 mL | 144.76 mL | 289.51 mL |
| 0.5 mM | 5.79 mL | 28.95 mL | 57.9 mL |
| 1 mM | 2.9 mL | 14.48 mL | 28.95 mL |
| 5 mM | 0.58 mL | 2.9 mL | 5.79 mL |
*The above data is based on the productmolecular weight 345.407. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A18338 |
|---|---|
| Actions | Agonist |
| CAS No. | 179756-58-2 |
| Formula | C16H23N7O2 |
| M. Wt | 345.407 |
| Purity | >98% |
| Synonyms | F11440, F 11440 |
| SMILES | O=C(N1C)N(CCCCN2CCN(C3=NC=CC=N3)CC2)N=CC1=O |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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