Fig. 1 · Structure
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ER121
ErbB2 Inhibitor
ER121 is a selective ErbB2 kinase inhibitor that exhibits oral bioavailability and non-toxic properties. It demonstrates potent antitumor activity, making it a valuable tool for the investigation of HER2-related breast cancer. Researchers can utilize ER121 to explore its effects on signaling pathways and evaluate potential therapeutic strategies in oncology.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2360839-74-1 |
| Applications | ErbB2 Inhibitor |
| Formula | C24H27ClFN5O3 |
| Molecular Weight | 487.95 |
| Synonyms | SGI-078 |
| SMILES | O=C(NC1=CC2=C(NC3=CC=C(C(Cl)=C3)F)N=CN=C2C=C1OCC)/C=C/CN(CCCO)C |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.