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Ersentilide

β1-adrenoceptor Antagonist

Ersentilide is a β1-adrenoceptor antagonist known for its effectiveness as an I_Kr blocker. This compound demonstrates significant antiarrhythmic properties in various intact animal models, making it a valuable tool for research in cardiovascular pharmacology and the study of arrhythmias. Its targeting of β1-adrenoceptors allows for the exploration of therapeutic interventions in cardiac conditions associated with dysregulated adrenergic signaling.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Antagonist
CAS Number	125279-79-0
Applications	β1-adrenoceptor Antagonist
Formula	C₂₁H₂₆N₄O₅S
Molecular Weight	446.52
SMILES	CS(NC(C=C1)=CC=C1OC[C@@H](O)CNCCOC2=CC=C(N3C=CN=C3)C=C2)(=O)=O

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.