Fig. 1 · Structure
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Fasitibant chloride
B2R Antagonist
Fasitibant chloride is a potent and selective nonpeptide antagonist of the bradykinin B2 receptor (B2R). It has demonstrated significant efficacy in reducing joint pain and alleviating joint edema in the Carrageenan-induced arthritis rat model. This compound is valuable for research in pain management and inflammation pathways.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 1157852-02-2 |
| Applications | B2R Antagonist |
| Formula | C36H49Cl3N6O6S |
| Molecular Weight | 800.23 |
| Synonyms | MEN16132 free base |
| SMILES | O=C(N(CC1)CCN1C([C@@H](N)CCC[N+](C)(C)C)=O)C2(CCOCC2)N[S](=O)(C(C=CC(Cl)=C3COC4=CC=CC(C(C)=C5)=C4N=C5C)=C3Cl)=O.[Cl-] |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.