Fig. 1 · Structure
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FK 453
Adenosine A1 Receptor Antagonist
FK 453 is a potent and selective antagonist of the adenosine A1 receptor, exhibiting an IC50 value of 17.2 nM. This compound plays a vital role in research related to cardiovascular and neuroprotective effects, making it a valuable tool for studies investigating adenosine signaling pathways. Its ability to inhibit A1 receptor activity provides insights into potential therapeutic applications in various biological contexts.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 121524-18-3 |
| Applications | Adenosine A1 Receptor Antagonist |
| Formula | C23H25N3O2 |
| Molecular Weight | 375.46 |
| SMILES | O=C(/C=C/C1=C2C=CC=CN2N=C1C3=CC=CC=C3)N4[C@@H](CCO)CCCC4 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.