FR 75513 is a 1,1'-biphenyl-2,6-dicarboxylic acid diester compound known for its ability to inhibit detrusor muscle contraction. It demonstrates significant pharmacological activity, with an IC50 of 3.3 μg/mL in guinea pig bladder assays and an ID50 of 0.04 mg/kg following intravenous administration in anesthetized rats. This compound is valuable for research applications in urology and muscle contraction studies.
FR 75513 is a 1,1'-biphenyl-2,6-dicarboxylic acid diester compound known for its ability to inhibit detrusor muscle contraction. It demonstrates significant pharmacological activity, with an IC50 of 3.3 μg/mL in guinea pig bladder assays and an ID50 of 0.04 mg/kg following intravenous administration in anesthetized rats. This compound is valuable for research applications in urology and muscle contraction studies.
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