Fig. 1 · Structure
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FXa-IN-1
FXa Inhibitor
FXa-IN-1 is a potent factor Xa (FXa) inhibitor, exhibiting an IC50 of 3 nM and a Ki value of 0.7 nM. This compound demonstrates notable oral bioavailability and a favorable half-life in vivo, making it effective for research in thromboembolic disorders. FXa-IN-1 is valuable for studying coagulation pathways and assessing therapeutic interventions in related diseases.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 441328-10-5 |
| Applications | FXa Inhibitor |
| Formula | C24H18F5N5O |
| Molecular Weight | 487.42 |
| SMILES | O=C(NC1=CC=C(C(N(C)C)=N)C=C1F)C2=CC(C(F)(F)F)=NN2C3=C(F)C=C(C=CC=C4)C4=C3 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.