G007-LK

Catalog No.: A15528

TNKS inhibitor

G007-LK Chemical Structure

CAS NO. 1380672-07-0

G007-LK displays high selectivity toward tankyrases 1 and 2 with biochemical IC50 values of 46 nM and 25 nM, respectively, and a cellular IC50 value of 50 nM combined with an excellent pharmacokinetic profile in mice,

Availability: In stock

Package Price Qty
5 mg

Regular Price: $80.00

Special Price $64.00

10 mg

Regular Price: $140.00

Special Price $112.00

25 mg

Regular Price: $300.00

Special Price $240.00

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

G007-LK displays high selectivity toward tankyrases 1 and 2 with biochemical IC50 values of 46 nM and 25 nM, respectively, and a cellular IC50 value of 50 nM combined with an excellent pharmacokinetic profile in mice,
Targets
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.87 mL 94.35 mL 188.69 mL
0.5 mM 3.77 mL 18.87 mL 37.74 mL
1 mM 1.89 mL 9.43 mL 18.87 mL
5 mM 0.38 mL 1.89 mL 3.77 mL

*The above data is based on the productmolecular weight 529.96. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15528
Actions Inhibitor
M. Wt 529.96
Formula C25H16ClN7O3S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1380672-07-0
Synonyms G007 LK, G007LK
SMILES CS(=O)(=O)C1=CN=C(C=C1)C2=NN=C(N2C3=CC=CC=C3Cl)C=CC4=NN=C(O4)C5=CC=C(C=C5)C#N

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