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Fig. 1 · Structure
Cat. No.
A56879
CAS No.
1663564-42-8
Formula
C25H28N4OS
Mol. Weight
432.59

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GAT100

Cannabinoid 1 Receptor Negative Allosteric Modulator

GAT100 is a negative allosteric modulator targeting the cannabinoid 1 receptor (CB1R). It functions by reducing the potency and efficacy of orthosteric CB1R agonists such as CP55,940, influencing key signaling pathways including β-arrestin 1 recruitment and ERK1/2 phosphorylation. GAT100 is a valuable tool for investigating the role of CB1R in psychobehavioral and somatic disorders, facilitating research on therapeutic strategies for conditions influenced by cannabinoid signaling.

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Specifications

Manufacturer Adooq Bioscience
Actions Modulator
CAS Number 1663564-42-8
Applications Cannabinoid 1 Receptor Negative Allosteric Modulator
Formula C25H28N4OS
Molecular Weight 432.59
SMILES
O=C(NCCC1=CC=C(C=C1)N2CCCCC2)C=3NC=4C=CC(N=C=S)=CC4C3CC

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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