Fig. 1 · Structure
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GAT211
CB1R PAM
GAT211 is a positive allosteric modulator of the cannabinoid 1 receptor (CB1R). It enhances cAMP and β-arrestin2 signaling with EC50 values of 260 nM and 650 nM, respectively. GAT211 is suitable for research focused on neuropathic and inflammatory pain pathways, making it a valuable tool for studying cannabinoid receptor modulation and its therapeutic implications.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Modulator |
| CAS Number | 102704-40-5 |
| Applications | CB1R PAM |
| Formula | C22H18N2O2 |
| Molecular Weight | 342.39 |
| SMILES | O=[N+]([O-])CC(C1=CC=CC=C1)C2=C(NC3=C2C=CC=C3)C4=CC=CC=C4 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.