Fig. 1 · Structure
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GBR-12879 methanesulfonate
Dopamine Transporter Inhibitor
GBR-12879 methanesulfonate is a selective inhibitor of the dopamine transporter (DAT), which regulates dopamine levels in the synaptic cleft. By blocking dopamine reuptake, it enhances dopaminergic transmission, making it valuable for studies of neuropharmacology and potential therapeutic applications in conditions like Parkinson's disease and mood disorders. Its activity in modulating dopamine signaling pathways provides insights into the mechanisms of action of various neurological treatments.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 77862-93-2 |
| Applications | Dopamine Transporter Inhibitor |
| Formula | C30H38F2N2O7S2 |
| Molecular Weight | 640.76 |
| SMILES | O=S(O)(C)=O.FC1=CC=C(C(C2=CC=C(C=C2)F)OCCN3CCN(CC3)C/C=C/C4=CC=CC=C4)C=C1.O=S(O)(C)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.