GG-818

Catalog No.: A58622
α1 Adrenoceptor Antagonist
GG-818 is a selective antagonist of the α1 adrenoceptor, exhibiting potent inhibition with pKi values of 9.7 for α1a, 7.8 for α1b, and 7.6 for α1d. This compound is valuable in the study of benign prostatic hyperplasia and contributes to understanding α1 adrenoceptor-mediated signaling pathways and their implications in urological health. Its specificity may facilitate research into potential therapeutic interventions targeting α1 adrenergic receptors.
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Adooq Products cited in reputable paper
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Biological Activity
DescriptionGG-818 is a selective antagonist of the α1 adrenoceptor, exhibiting potent inhibition with pKi values of 9.7 for α1a, 7.8 for α1b, and 7.6 for α1d. This compound is valuable in the study of benign prostatic hyperplasia and contributes to understanding α1 adrenoceptor-mediated signaling pathways and their implications in urological health. Its specificity may facilitate research into potential therapeutic interventions targeting α1 adrenergic receptors.
Product Information
Catalog NumA58622
FormulaC26H29F4N3O5S
Molecular Weight571.58
CAS Number179535-60-5
SMILESO=S(C1=CC(CCN2CCC(C3=NC(COCC(F)(F)F)=C(C4=CC=C(F)C=C4)O3)CC2)=CC=C1OC)(N)=O
SynonymsGW 1818
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