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GIPR antagonist 1

GIPR Antagonist

GIPR Antagonist 1 is a potent inhibitor of the glucose-dependent insulinotropic polypeptide receptor (GIPR) with an IC50 of 4.8 nM. By effectively blocking GIPR signaling, this compound serves as a valuable tool in the study of type 2 diabetes and obesity. Its ability to modulate GIPR activity makes it significant for research focused on glucose metabolism and insulin regulation.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Inhibitor
CAS Number	3059497-30-9
Applications	GIPR Antagonist
Formula	C₂₈H₂₉FN₄O₄
Molecular Weight	504.55
SMILES	FC(C=C1NC(N2[C@H](CCC2)C(NC3=CC=C(C4=C(N=C(C=C4)C(O)=O)C)C=C3)=O)=O)=C(C=C1)C(C)C

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.