Fig. 1 · Structure
Documents & Downloads
GK241
GK241 is a 2-oxoamide-based compound that selectively inhibits human and mouse group IIA secretory phospholipase A2 (GIIA sPLA2), with IC50 values of 143 nM and 68 nM, respectively. The compound has been examined for its inhibitory mechanism through molecular dynamics simulations. GK241 serves as a valuable tool for exploring the biochemical pathways involving phospholipase A2 and its role in various biological processes.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| CAS Number | 1899930-93-8 |
| Formula | C21H39NO4 |
| Molecular Weight | 369.54 |
| SMILES | CCCCCCCCCCCCCCC(C(N[C@H](C(O)=O)C(C)C)=O)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.