Catalog No.: A21466

FFA2/GPR43 antagonist


GLPG0974 Chemical Structure

CAS NO. 1391076-61-1

GLPG0974 is a free fatty acid receptor-2 (FFA2/GPR43) antagonist with an IC50 of 9 nM.

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Biological Activity

GLPG0974 is a free fatty acid receptor-2 (FFA2/GPR43) antagonist with an IC50 of 9 nM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.62 mL 103.09 mL 206.19 mL
0.5 mM 4.12 mL 20.62 mL 41.24 mL
1 mM 2.06 mL 10.31 mL 20.62 mL
5 mM 0.41 mL 2.06 mL 4.12 mL

*The above data is based on the productmolecular weight 485. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21466
Actions Antagonist
CAS No. 1391076-61-1
Formula C25H25ClN2O4S
M. Wt 485
Solubility DMSO
Purity >98%
Synonyms GLPG 0974, GLPG-0974
SMILES O=C(O)CCCN(C([[email protected]]1(C)N(C(C2=CSC3=CC=CC=C32)=O)CC1)=O)CC4=CC=CC(Cl)=C4

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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