Biological Activity
GLPG0974 is a free fatty acid receptor-2 (FFA2/GPR43) antagonist with an IC50 of 9 nM.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 20.62 mL | 103.09 mL | 206.19 mL |
0.5 mM | 4.12 mL | 20.62 mL | 41.24 mL |
1 mM | 2.06 mL | 10.31 mL | 20.62 mL |
5 mM | 0.41 mL | 2.06 mL | 4.12 mL |
*The above data is based on the productmolecular weight 485. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A21466 |
---|---|
Actions | Antagonist |
CAS No. | 1391076-61-1 |
Formula | C25H25ClN2O4S |
M. Wt | 485 |
Solubility | DMSO |
Purity | >98% |
Synonyms | GLPG 0974, GLPG-0974 |
SMILES | O=C(O)CCCN(C([[email protected]]1(C)N(C(C2=CSC3=CC=CC=C32)=O)CC1)=O)CC4=CC=CC(Cl)=C4 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
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