Fig. 1 · Structure
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GluN1/3A-IN-1
GluN1/GluN3A Inhibitor
GluN1/3A-IN-1 is a potent inhibitor of the GluN1/GluN3A NMDA receptors, with an IC50 value of 0.98 µM. This compound exerts its inhibitory effects by targeting the pre-M1 region and forming hydrogen bond interactions with critical residues within the receptor. GluN1/3A-IN-1 is primarily utilized in research focused on neurological diseases linked to GluN1 and GluN3A receptor dysregulation, providing valuable insights into potential therapeutic strategies.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 1147526-22-4 |
| Applications | GluN1/GluN3A Inhibitor |
| Formula | C23H17NO5 |
| Molecular Weight | 387.38 |
| SMILES | O=C(C1=C(C=C(C=C1)O)O)OCC(C2C(C3=CC=CC=C3)=NC4=C2C=CC=C4)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.