Fig. 1 · Structure
Documents & Downloads
GNE-235
Furan Ring Analogue
GNE-235 is a furan ring analogue that selectively targets the second bromodomain of PBRM1, exhibiting a binding affinity (KD) of 0.28 ± 0.02 μM. This compound serves as a valuable tool for investigating the cellular functions of PBRM1, contributing to the understanding of its role in various biological processes and potential therapeutic applications.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| CAS Number | 3036574-72-5 |
| Applications | Furan Ring Analogue |
| Formula | C13H16N4O |
| Molecular Weight | 244.29 |
| SMILES | C[C@H]1CCCN1C2=C(N)N=NC(C3=CC=CO3)=C2 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.