GnRH-R antagonist 1 is a potent GnRH receptor antagonist that exhibits high binding affinity with an IC50 of 0.57 nM and strong in vitro antagonistic activity at an IC50 of 2.18 nM. This compound is membrane-permeable and orally bioavailable, making it suitable for various research applications. It is particularly valuable in studies focused on advanced prostate cancer and in investigating the prevention of premature luteinizing hormone peaks.
GnRH-R antagonist 1 is a potent GnRH receptor antagonist that exhibits high binding affinity with an IC50 of 0.57 nM and strong in vitro antagonistic activity at an IC50 of 2.18 nM. This compound is membrane-permeable and orally bioavailable, making it suitable for various research applications. It is particularly valuable in studies focused on advanced prostate cancer and in investigating the prevention of premature luteinizing hormone peaks.
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