Fig. 1 · Structure
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GR125487 sulfamate
5-HT4 Receptor Antagonist
GR125487 sulfamate is a selective antagonist of the 5-HT4 receptor, which plays a significant role in various cognitive and gastrointestinal functions. This compound effectively inhibits cognitive enhancement, making it valuable for researching memory disorders, mood disorders, gastrointestinal dysfunctions, and urinary tract issues. Its oral bioactivity allows for convenient administration in preclinical studies.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 859502-43-5 |
| Applications | 5-HT4 Receptor Antagonist |
| Formula | C19H29FN4O8S2 |
| Molecular Weight | 524.58 |
| SMILES | O=C(C1=C(NC2=C1C=C(F)C=C2)OC)OCC3CCN(CC3)CCNS(=O)(C)=O.O=S(O)(N)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.