Target & Activity
| Target | Activity | Value |
|---|---|---|
| GRP94 | IC50 | 2 nM |
Fig. 1 · Structure
Documents & Downloads
Grp94 Inhibitor-1
Cat. No.
A20073
CAS
2234897-35-7
Grp94 inhibitor
Grp94 Inhibitor-1 is a potent, selective Grp94 inhibitor with an IC50 value of 2 nM, and over 1000-fold selectivity to Grp94 against Hsp90α.
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Biological Activity
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2234897-35-7 |
| Applications | Grp94 inhibitor |
| Formula | C22H28N2O2 |
| Molecular Weight | 352.47 |
| SMILES | O=C(C1=CC(C2=CC=C(C(C)C)C=C2)=CC=C1N[C@H]3CC[C@H](O)CC3)N |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.