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GRPR antagonist-2

GRPR Antagonist

GRPR Antagonist-2 is a potent antagonist of the gastrin-releasing peptide receptor (GRPR), demonstrating cytotoxic effects against specific cancer cell lines, with IC50 values of 0.77 μM in HGC-27 cells and 2.5 μM in Pan02 cells. This compound is primarily employed in anticancer research to explore GRPR-mediated signaling pathways and their implications in tumor growth and progression.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Antagonist
CAS Number	3052544-42-7
Applications	GRPR Antagonist
Formula	C₂₈H₃₂F₃N₅O₄
Molecular Weight	559.58
SMILES	CC(C)(OC(N1CCN(CC1)C([C@H](CC2=CNC3=C2C=CC=C3)NC(NC4=CC=C(C=C4)C(F)(F)F)=O)=O)=O)C

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.