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GRPR antagonist-3

GRPR Antagonist

GRPR antagonist-3 targets the gastrin-releasing peptide receptor (GRPR) and demonstrates potent antagonistic activity with an IC50 of 121 nM. This compound exhibits stability in rat plasma and is resistant to microsomal oxidative metabolism in vitro. GRPR antagonist-3 can be radiolabeled with fluorine-18, making it suitable for positron emission tomography (PET) imaging applications in preclinical studies and cancer research.

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Specifications

Manufacturer	Adooq Bioscience
CAS Number	2077238-49-2
Applications	GRPR Antagonist
Formula	C₃₃H₃₇FN₆O₅
Molecular Weight	616.68
SMILES	O=C(NC1=CC=C(C=C1)[N+]([O-])=O)N[C@](CC2=CNC3=CC=CC=C23)(C)C(NCC4(C5=CC=C(C=N5)OCCF)CCCCC4)=O

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.