GS967

Catalog No.: A14361

late INa Inhibitor

GS967

GS967 Chemical Structure

CAS NO. 1262618-39-2

GS967 is a novel, potent, and selective inhibitor of cardiac late sodium current(late INa); inhibits ATX-II-induced late I(Na) in ventricular myocytes and isolated hearts with IC(50) values of 0.13 and 0.21 uM, respectively.

Availability: In stock

Package Price Qty
5 mg
$50.00
10 mg
$85.00
25 mg
$150.00
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Biological Activity

GS967 is a novel, potent, and selective inhibitor of cardiac late sodium current(late INa); inhibits ATX-II-induced late I(Na) in ventricular myocytes and isolated hearts with IC(50) values of 0.13 and 0.21 uM, respectively.
In vitro DMSO 38 mg/mL (109.44 mM)
Water Insoluble
Ethanol 39 mg/mL (112.32 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 28.8 mL 144 mL 288 mL
0.5 mM 5.76 mL 28.8 mL 57.6 mL
1 mM 2.88 mL 14.4 mL 28.8 mL
5 mM 0.58 mL 2.88 mL 5.76 mL

*The above data is based on the productmolecular weight 347.22. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A14361
Actions Inhibitor
CAS No. 1262618-39-2
Formula C14H7F6N3O
M. Wt 347.22
Purity >98%
Synonyms GS-967, GS 967
SMILES FC(F)(F)C1=NN=C2C=CC(C3=CC=C(OC(F)(F)F)C=C3)=CN21
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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