Biological Activity
GS967 is a novel, potent, and selective inhibitor of cardiac late sodium current(late INa); inhibits ATX-II-induced late I(Na) in ventricular myocytes and isolated hearts with IC(50) values of 0.13 and 0.21 uM, respectively.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 28.8 mL | 144 mL | 288 mL |
0.5 mM | 5.76 mL | 28.8 mL | 57.6 mL |
1 mM | 2.88 mL | 14.4 mL | 28.8 mL |
5 mM | 0.58 mL | 2.88 mL | 5.76 mL |
*The above data is based on the productmolecular weight 347.22. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A14361 |
---|---|
Actions | Inhibitor |
M. Wt | 347.22 |
Formula | C14H7F6N3O |
Solubility | DMSO |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 1262618-39-2 |
Synonyms | GS-967, GS 967 |
SMILES | FC(F)(F)C1=NN=C2C=CC(C3=CC=C(OC(F)(F)F)C=C3)=CN21 |
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