GSK1070916

Catalog No.: A11168
Aurora Kinase B/C inhibitor

GSK1070916 is a potent Aurora B/C kinase inhibitor (with IC50 of 3.5 nM/6.5 nM) with broad antitumor activity in tissue culture cells and human tumor xenograft models.

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Product Name Price Stock Qty
GSK1070916 5mg
Special Price $72.00 Regular Price $90.00
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GSK1070916 10mg
Special Price $120.00 Regular Price $150.00
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GSK1070916 50mg
Special Price $320.00 Regular Price $400.00
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GSK1070916 100mg
Special Price $560.00 Regular Price $700.00
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GSK1070916 10mM * 1mL in DMSO
Special Price $80.00 Regular Price $100.00
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Biological Activity
Discription

GSK1070916 is a potent Aurora B/C kinase inhibitor (with IC50 of 3.5 nM/6.5 nM) with broad antitumor activity in tissue culture cells and human tumor xenograft models.

Targets
Target Value
Product Information
Catalog Num A11168
Formula C30H33N7O
Molecular Weight 507.63
CAS Number 942918-07-2
SMILES CCN1C=C(C(=N1)C2=CC=C(C=C2)NC(=O)N(C)C)C3=C4C=C(NC4=NC=C3)C5=CC(=CC=C5)CN(C)C
Synonyms GSK-1070916
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro (25°C) DMSO 91 mg/mL (179.26 mM)
Water Insoluble
Ethanol 8 mg/mL (15.75 mM)
In vivo 2% Cremophor EL, 2% N,N-dimethylacetamide, pH 5.0 28 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.7 mL 98.5 mL 196.99 mL
0.5 mM 3.94 mL 19.7 mL 39.4 mL
1 mM 1.97 mL 9.85 mL 19.7 mL
5 mM 0.39 mL 1.97 mL 3.94 mL
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

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