Fig. 1 · Structure
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GSK239512
H3 Receptor Antagonist
GSK239512 is a potent antagonist of the histamine H3 receptor, demonstrating effective central nervous system penetration. This compound is primarily utilized in research investigating mild-to-moderate Alzheimer's disease (AD) and may provide insights into therapeutic strategies targeting cognitive impairment associated with this condition.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 720691-69-0 |
| Applications | H3 Receptor Antagonist |
| Formula | C23H27N3O2 |
| Molecular Weight | 377.48 |
| SMILES | O=C1N(C2=CC=C(OC3=CC=C4CCN(C5CCC5)CCC4=C3)N=C2)CCC1 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.