GSK2636771

Catalog No.: A11784

PI3K Inhibitor

GSK2636771

GSK2636771 Chemical Structure

CAS NO. 1372540-25-4

GSK2636771 is a potent, orally bioavailable, PI3K beta-selective inhibitor.

Availability: In stock

Package Price Qty
5 mg
$70.00
10 mg
$120.00
50 mg
$350.00
100 mg
$550.00
10mM * 1mL in DMSO
$80.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.
  • Pridham KJ, .et al. PIK3CB/p110β is a selective survival factor for glioblastoma, Neuro Oncol, 2018, Mar 27;20(4):494-505 PMID: 29016844

Biological Activity

GSK2636771 is a potent, orally bioavailable, PI3K beta-selective inhibitor.
Targets
PI3Kβ
In vitro DMSO 28 mg/mL (64.6 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.07 mL 115.37 mL 230.73 mL
0.5 mM 4.61 mL 23.07 mL 46.15 mL
1 mM 2.31 mL 11.54 mL 23.07 mL
5 mM 0.46 mL 2.31 mL 4.61 mL

*The above data is based on the productmolecular weight 433.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11784
Actions Inhibitor
CAS No. 1372540-25-4
Formula C22H22F3N3O3
M. Wt 433.4
Solubility DMSO
Purity >98%
Synonyms GSK 2636771
SMILES CC1=C(C=CC=C1C(F)(F)F)CN2C(=NC3=C2C=C(C=C3C(=O)O)N4CCOCC4)C
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy GSK2636771 | GSK2636771 Supplier | purchase | cost | manufacturer | order | distributor | buy 1372540-25-4| 1372540-25-4 Supplier | purchase 1372540-25-4 | 1372540-25-4 cost | 1372540-25-4 manufacturer | order 1372540-25-4 | 1372540-25-4 distributor
Rewards