Fig. 1 · Structure
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GSK264220A
Endothelial Lipase Inhibitor
GSK264220A is a selective inhibitor of endothelial lipase, exhibiting an IC50 value of 16 nM. This compound plays a crucial role in modulating lipid metabolism and has potential applications in cardiovascular disease research by reducing endothelial lipase activity, thereby potentially lowering lipid levels and associated cardiovascular risks.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 685506-42-7 |
| Applications | Endothelial Lipase Inhibitor |
| Formula | C17H21N3O4S |
| Molecular Weight | 363.43 |
| SMILES | O=C(NC1=C(C)OC(S(=O)(N2CCCCC2)=O)=C1)NC3=CC=CC=C3 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.