GSK2801

Catalog No.: A14015

BAZ2A and BAZ2B inhibitor

GSK2801

GSK2801 Chemical Structure

CAS NO. 1619994-68-1

GSK2801 is a very potent inhibitor of the BAZ2 family of bromodomain containing proteins

Availability: In stock

Package Price Qty
10 mg
$70.00
25 mg
$140.00
50 mg
$220.00
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Biological Activity

GSK2801 is a very potent inhibitor of the BAZ2 family of bromodomain containing proteins
Targets
BAZ2B BAZ2A
136 nM(Kd)257 nM(Kd)
In vitro (25°C) DMSO Warmed: 67 mg/mL (180.37 mM)
Water Insoluble
Ethanol Warmed: 6 mg/mL (16.15 mM)
In vivo 0.5% CMC+1% Tween 80 28 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 26.92 mL 134.58 mL 269.15 mL
0.5 mM 5.38 mL 26.92 mL 53.83 mL
1 mM 2.69 mL 13.46 mL 26.92 mL
5 mM 0.54 mL 2.69 mL 5.38 mL

*The above data is based on the productmolecular weight 371.54. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A14015
Actions Inhibitor
CAS No. 1619994-68-1
Formula C20H21NO4S
M. Wt 371.54
Purity >98%
Synonyms GSK-2801, GSK 2801
SMILES CCCOC1=CC2=C(C=C(N2C=C1)C(=O)C)C3=CC=CC=C3S(=O)(=O)C
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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