Catalog No.: A14015

BAZ2A and BAZ2B inhibitor


GSK2801 Chemical Structure

CAS NO. 1619994-68-1

GSK2801 is a very potent inhibitor of the BAZ2 family of bromodomain containing proteins

Availability: In stock

Package Price Qty
10 mg
25 mg
50 mg
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

GSK2801 is a very potent inhibitor of the BAZ2 family of bromodomain containing proteins
136 nM(Kd)257 nM(Kd)
In vitro (25°C) DMSO Warmed: 67 mg/mL (180.37 mM)
Water Insoluble
Ethanol Warmed: 6 mg/mL (16.15 mM)
In vivo 0.5% CMC+1% Tween 80 28 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 26.92 mL 134.58 mL 269.15 mL
0.5 mM 5.38 mL 26.92 mL 53.83 mL
1 mM 2.69 mL 13.46 mL 26.92 mL
5 mM 0.54 mL 2.69 mL 5.38 mL

*The above data is based on the productmolecular weight 371.54. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A14015
Actions Inhibitor
CAS No. 1619994-68-1
Formula C20H21NO4S
M. Wt 371.54
Purity >98%
Synonyms GSK-2801, GSK 2801

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy GSK2801 | GSK2801 Supplier | purchase | cost | manufacturer | order | distributor | buy 1619994-68-1| 1619994-68-1 Supplier | purchase 1619994-68-1 | 1619994-68-1 cost | 1619994-68-1 manufacturer | order 1619994-68-1 | 1619994-68-1 distributor