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$0.00 Biological Activity
GSK2801 is a very potent inhibitor of the BAZ2 family of bromodomain containing proteins
Targets
| BAZ2B | BAZ2A | |||
| 136 nM(Kd) | 257 nM(Kd) |
| In vitro (25°C) | DMSO | Warmed: 67 mg/mL (180.37 mM) | |
| Water | Insoluble | ||
| Ethanol | Warmed: 6 mg/mL (16.15 mM) | ||
| In vivo | 0.5% CMC+1% Tween 80 | 28 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 26.92 mL | 134.58 mL | 269.15 mL |
| 0.5 mM | 5.38 mL | 26.92 mL | 53.83 mL |
| 1 mM | 2.69 mL | 13.46 mL | 26.92 mL |
| 5 mM | 0.54 mL | 2.69 mL | 5.38 mL |
*The above data is based on the productmolecular weight 371.54. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A14015 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 1619994-68-1 |
| Formula | C20H21NO4S |
| M. Wt | 371.54 |
| Purity | >98% |
| Synonyms | GSK-2801, GSK 2801 |
| SMILES | CCCOC1=CC2=C(C=C(N2C=C1)C(=O)C)C3=CC=CC=C3S(=O)(=O)C |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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