GSK2807 Trifluoroacetate

Catalog No.: A21731

SMYD3 inhibitor

GSK2807 Trifluoroacetate

GSK2807 Trifluoroacetate Chemical Structure

CAS NO. 2245255-66-5

GSK2807 Trifluoroacetate is a potent, selective and SAM-competitive inhibitor of SMYD3, with a Ki of 14 nM and an IC50 of 130 nM.

Availability: In stock

Package Price Qty
5 mg
$225.00
10 mg
$388.00
50 mg
$1,150.00
100 mg
$2,300.00
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Biological Activity

GSK2807 Trifluoroacetate is a potent, selective and SAM-competitive inhibitor of SMYD3, with a Ki of 14 nM and an IC50 of 130 nM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.65 mL 88.26 mL 176.51 mL
0.5 mM 3.53 mL 17.65 mL 35.3 mL
1 mM 1.77 mL 8.83 mL 17.65 mL
5 mM 0.35 mL 1.77 mL 3.53 mL

*The above data is based on the productmolecular weight 566.53. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21731
Actions Inhibitor
CAS No. 2245255-66-5
Formula C21H33F3N8O7
M. Wt 566.53
Solubility DMSO
Purity >98%
Synonyms GSK 2807, GSK-2807
SMILES NC1=C2C(N([[email protected]]3[[email protected]](O)[[email protected]](O)[[email protected]@H](CN(CC[[email protected]](N)C(O)=O)CCCN(C)C)O3)C=N2)=NC=N1.OC(C(F)(F)F)=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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