GSK2982772

Catalog No.: A19380

RIP1 kinase inhibitor

GSK2982772

GSK2982772 Chemical Structure

CAS NO. 1622848-92-3

GSK2982772 is a potent, orally active and ATP competitive RIP1 kinase inhibitor with IC50 values of 16 nM and 20 nM for human and monkey RIP1, respectively.

Availability: In stock

Package Price Qty
1 mg
$70.00
5 mg
$160.00
10 mg
$250.00
50 mg
$720.00
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Biological Activity

GSK2982772 is a potent, orally active and ATP competitive RIP1 kinase inhibitor with IC50 values of 16 nM and 20 nM for human and monkey RIP1, respectively.
In vitro DMSO 66 mg/mL (174.87 mM)
Water Insoluble
Ethanol 26 mg/mL (68.89 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 26.5 mL 132.49 mL 264.97 mL
0.5 mM 5.3 mL 26.5 mL 52.99 mL
1 mM 2.65 mL 13.25 mL 26.5 mL
5 mM 0.53 mL 2.65 mL 5.3 mL

*The above data is based on the productmolecular weight 377.4. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A19380
Actions Inhibitor
CAS No. 1622848-92-3
Formula C20H19N5O3
M. Wt 377.4
Purity >98%
Synonyms GSK 2982772, GSK 2982772
SMILES O=C(C1=NC(CC2=CC=CC=C2)=NN1)N[[email protected]]3COC4=CC=CC=C4N(C)C3=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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