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GSK4716

Catalog No.: A16956

ERRβ & ERRγ Agonist

GSK4716

GSK4716 Chemical Structure

CAS NO. 101574-65-6

GSK4716 is an Estrogen-related receptors ERRβ and ERRγ agonist with minimal activity for ERRα, ERα and ERβ

Availability: In stock

Package Price Qty
10 mg
$60.00
25 mg
$120.00
50 mg
$300.00
100 mg
$520.00
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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.
  • Sen He, .et al. The potential endocrine disruption mechanism of anthelmintic drug niclosamide by activating estrogen receptors and estrogen-related receptors, Toxicology, 2021, May 4;457:152805 PMID: 33961950

Biological Activity

GSK4716 is an Estrogen-related receptors ERRβ and ERRγ agonist with minimal activity for ERRα, ERα and ERβ
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 35.42 mL 177.09 mL 354.18 mL
0.5 mM 7.08 mL 35.42 mL 70.84 mL
1 mM 3.54 mL 17.71 mL 35.42 mL
5 mM 0.71 mL 3.54 mL 7.08 mL

*The above data is based on the productmolecular weight 282.34. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16956
Actions Agonist
CAS No. 101574-65-6
Formula C17H18N2O2
M. Wt 282.34
Purity >98%
Synonyms GSK 4716, GSK-4716, GW4716, GW 4716, GW-4716
SMILES O=C(N/N=C/C1=CC=C(C(C)C)C=C1)C2=CC=C(O)C=C2
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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