GSK6853

Catalog No.: A16330

BRPF1 bromodomain inhibitor

GSK6853

GSK6853 Chemical Structure

CAS NO. 1910124-24-1

GSK6853 is a potent and selective inhibitor of the BRPF1 bromodomain. shows excellent BRPF1 potency (pKd 9.5) and greater than 1600-fold selectivity over all other bromodomains tested.

Availability: In stock

Package Price Qty
5 mg
$80.00
10 mg
$140.00
50 mg
$420.00
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Biological Activity

GSK6853 is a potent and selective inhibitor of the BRPF1 bromodomain. shows excellent BRPF1 potency (pKd 9.5) and greater than 1600-fold selectivity over all other bromodomains tested.
In vitro DMSO Warmed: 77 mg/mL (188.04 mM)
Water Insoluble
Ethanol Warmed: 77 mg/mL (188.04 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.42 mL 122.11 mL 244.21 mL
0.5 mM 4.88 mL 24.42 mL 48.84 mL
1 mM 2.44 mL 12.21 mL 24.42 mL
5 mM 0.49 mL 2.44 mL 4.88 mL

*The above data is based on the productmolecular weight 409.48. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16330
Actions Inhibitor
CAS No. 1910124-24-1
Formula C22H27N5O3
M. Wt 409.48
Solubility DMSO
Purity >98%
Synonyms GSK-6853, GSK 6853
SMILES O=C(NC1=C(N2[[email protected]](C)CNCC2)C=C(N3C)C(N(C)C3=O)=C1)C4=CC=CC=C4OC
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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