GSK6853
Important Notice: For research use only. We do not sell to patients.
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Important Notice: For research use only. We do not sell to patients.
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Discription | GSK6853 is a potent and selective inhibitor of the BRPF1 bromodomain. shows excellent BRPF1 potency (pKd 9.5) and greater than 1600-fold selectivity over all other bromodomains tested. |
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Catalog Num | A16330 |
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Formula | C22H27N5O3 |
Molecular Weight | 409.48 |
CAS Number | 1910124-24-1 |
SMILES | O=C(NC1=C(N2[C@H](C)CNCC2)C=C(N3C)C(N(C)C3=O)=C1)C4=CC=CC=C4OC |
Synonyms | GSK-6853, GSK 6853 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | Warmed: 77 mg/mL (188.04 mM) | |
Water | Insoluble | ||
Ethanol | Warmed: 77 mg/mL (188.04 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 24.42 mL | 122.11 mL | 244.21 mL |
0.5 mM | 4.88 mL | 24.42 mL | 48.84 mL |
1 mM | 2.44 mL | 12.21 mL | 24.42 mL |
5 mM | 0.49 mL | 2.44 mL | 4.88 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2