Fig. 1 · Structure
Documents & Downloads
GSK789
BD1 Inhibitor
GSK789 is a highly selective inhibitor targeting the first bromodomain (BD1) of the BET family. This compound exhibits potent antitumor and immunomodulatory activities, making it a valuable tool for investigating therapeutic strategies in cancer treatment and immune response modulation. GSK789's cell-permeable properties enhance its usability in various biological research applications.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2540591-06-6 |
| Applications | BD1 Inhibitor |
| Formula | C26H33N5O3 |
| Molecular Weight | 463.57 |
| SMILES | O=C([C@@H]1CN(C)CC[C@H]1NC2=C3NC(C(C)=CC3=C(C4=CC=CO4)C=N2)=O)NC5CCCCC5 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.