GSK864

Name: GSK864
Brand: Adooq Bioscience
SKU: A20737
Rating: 5 (288 reviews)

Catalog No.: A20737

IDH1 mutant inhibitor

GSK864 is an isocitrate dehydrogenase 1 (IDH1) mutant inhibitor; inhibits IDH1 mutants R132C, R132H, and R132G with IC50 values of 8.8, 15.2 and 16.6 nM.

Skip to the end of the images gallery

GSK864 1816331-66-4 IDH1 mutant inhibitor

Skip to the beginning of the images gallery

Grouped product items
Size	Price	Stock
1mg	$60.00	In stock
5mg	$155.00	In stock
10mg	$285.00	In stock
25mg	$570.00	In stock
50mg	$915.00	In stock
100mg	$1,475.00	In stock
*10mM 1mL in DMSO**	$190.00	In stock
Bulk Size	Bulk Discount

Bulk Inquiry

Notify me when the price drops

Free Delivery on orders over $500

Research use only. We do not sell to patients.

Data Sheet SDS

Loading distributor info...

Adooq Products cited in reputable paper

Biological Activity

Description	GSK864 is an isocitrate dehydrogenase 1 (IDH1) mutant inhibitor; inhibits IDH1 mutants R132C, R132H, and R132G with IC50 values of 8.8, 15.2 and 16.6 nM.

Product Information

Catalog Num	A20737
Formula	C30H31FN6O4
Molecular Weight	558.6
CAS Number	1816331-66-4
SMILES	FC(C=C1)=CC=C1CN2N=C(C(NC3=CC(C)=C(OC)C(C)=C3)=O)C4=C2[C@](C(N)=O)(C)CN(C(C5=CC=CN5)=O)C4
Synonyms	GSK 864, GSK-864
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

* Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C₁V₁ = C₂V₂