Fig. 1 · Structure
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H4R antagonist 2
H4R Antagonist
H4R Antagonist 2 is a potent antagonist of the histamine H4 receptor (H4R), a Furo[3,2-d]pyrimidine derivative. This compound exhibits significant biological activity in modulating immune responses and is primarily utilized in research focused on rheumatoid arthritis and other inflammatory conditions. Its effectiveness in H4R antagonism makes it a valuable tool for investigating the therapeutic potential in various pathologies related to immune system dysregulation.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 1148115-99-4 |
| Applications | H4R Antagonist |
| Formula | C13H17N5O |
| Molecular Weight | 259.31 |
| SMILES | NC1=NC(N2CC(NC)C2)=C(OC3=C4CCC3)C4=N1 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.