Fig. 1 · Structure
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hMC1R agonist 1
hMC1R Agonist
hMC1R Agonist 1 selectively activates the human melanocortin 1 receptor (hMC1R) with an EC50 of 3 nM. This compound demonstrates over 300-fold selectivity for hMC1R compared to hMC3R, hMC4R, and hMC5R, which have significantly higher EC50 values (902 nM, 915 nM, and >1000 nM, respectively). hMC1R Agonist 1 holds promise for potential therapeutic applications within the melanocortin receptor family, particularly in conditions related to pigmentation and metabolic regulation.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 3028881-87-7 |
| Applications | hMC1R Agonist |
| Formula | C54H70N14O8S2 |
| Molecular Weight | 1107.35 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.