hMC1R Agonist 1 selectively activates the human melanocortin 1 receptor (hMC1R) with an EC50 of 3 nM. This compound demonstrates over 300-fold selectivity for hMC1R compared to hMC3R, hMC4R, and hMC5R, which have significantly higher EC50 values (902 nM, 915 nM, and >1000 nM, respectively). hMC1R Agonist 1 holds promise for potential therapeutic applications within the melanocortin receptor family, particularly in conditions related to pigmentation and metabolic regulation.
hMC1R Agonist 1 selectively activates the human melanocortin 1 receptor (hMC1R) with an EC50 of 3 nM. This compound demonstrates over 300-fold selectivity for hMC1R compared to hMC3R, hMC4R, and hMC5R, which have significantly higher EC50 values (902 nM, 915 nM, and >1000 nM, respectively). hMC1R Agonist 1 holds promise for potential therapeutic applications within the melanocortin receptor family, particularly in conditions related to pigmentation and metabolic regulation.
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