Fig. 1 · Structure
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HY-078020
H1R Antagonist
HY-078020 is a selective antagonist of the histamine H1 receptor, demonstrating an IC50 value of 24.12 nM. This compound exhibits significant anti-inflammatory activity, making it a valuable tool for research into allergic diseases and related disorders. Its oral bioavailability enhances its potential for therapeutic applications in inflammatory conditions.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 2756222-90-7 |
| Applications | H1R Antagonist |
| Formula | C32H35ClN2O2 |
| Molecular Weight | 515.09 |
| SMILES | ClC(C=C1)=CC(CCC2=C/3N=CC=C2)=C1C3=C4CCN(CCCC5=CC(C(C)(C(O)=O)C)=CC=C5)CC/4 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.