Fig. 1 · Structure
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IACS-9571 TFA
Epigenetic Reader Domain Inhibitor
IACS-9571 TFA is a potent and selective inhibitor of the epigenetic reader domains TRIM24 and BRPF1, with an IC50 value of 8 nM for TRIM24 and Kd values of 31 nM and 14 nM for TRIM24 and BRPF1, respectively. This compound is valuable in research focusing on the modulation of epigenetic processes and gene expression regulation. Its specificity makes it a useful tool for investigating the roles of TRIM24 and BRPF1 in various biological contexts, including cancer and other diseases related to epigenetic dysregulation.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 1883598-69-3 |
| Applications | Epigenetic Reader Domain Inhibitor |
| Formula | C34H43F3N4O10S |
| Molecular Weight | 756.79 |
| Synonyms | ASIS-P040 TFA |
| SMILES | O=S(C1=CC=C(OC)C(OC)=C1)(NC2=C(OC3=CC(OCCC)=CC(OCCCCN(C)C)=C3)C=C(N4C)C(N(C)C4=O)=C2)=O.FC(F)(C(O)=O)F |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.