Fig. 1 · Structure
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ID110460002
Opioid Receptor Agonist
ID110460002 is a powerful agonist of the μ-opioid receptor (OPRM) and also engages the δ-opioid receptor (OPRD). It demonstrates robust activity through G protein signaling pathways at both receptors while showing minimal partial agonist activity towards the β-arrestin-2 pathway. The compound’s high intrinsic activity at OPRM remains consistent regardless of receptor expression levels, whereas its efficacy at OPRD is influenced by expression levels. ID110460002 is essential for research into pain mechanisms and analgesic responses, offering significant insights into opioid receptor function.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 1172882-21-1 |
| Applications | Opioid Receptor Agonist |
| Formula | C20H25FN4O |
| Molecular Weight | 356.45 |
| SMILES | O=C(NC1=CC=C(F)C=C1)NCC(C2=CC=C3C(=C2)CCN3C)N(C)C |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.