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Catalog No.: A11076

Opioid Receptor antagonist


JTC-801 Chemical Structure

CAS NO. 244218-51-7

JTC-801 is a selective antagonist for the nociceptin receptor, also known as the ORL-1 receptor.

Availability: In stock

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5 mg
10 mg
50 mg
100 mg
10mM * 1mL in DMSO
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  • Lihao Gu, .et al. 10-Hydroxy-2-Decenoic Acid in Royal Jelly Extract Induced Both Filaggrin and Amino Acid in a Cultured Human Three-Dimensional Epidermis Model, Cosmetics, 2017, 4(4), 48
  • Toshio Yawata, .et al. Brain opioid and nociceptin receptors are involved in regulation of bombesin-induced activation of central sympatho-adrenomedullary outflow in the rat, Mol Cell Biochem, 2016, Jan;411(1-2):201-11 PMID: 26427671

Biological Activity

JTC-801 is a selective antagonist for the nociceptin receptor, also known as the ORL-1 receptor.
In vitro (25°C) DMSO 88 mg/mL (196.45 mM)
Water Insoluble
Ethanol 30 mg/mL (66.97 mM)
In vivo 0.5% methylcellulose 28 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.32 mL 111.61 mL 223.21 mL
0.5 mM 4.46 mL 22.32 mL 44.64 mL
1 mM 2.23 mL 11.16 mL 22.32 mL
5 mM 0.45 mL 2.23 mL 4.46 mL

*The above data is based on the productmolecular weight 448. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11076
Actions Antagonist
CAS No. 244218-51-7
Formula C26H25N3O2.HCl
M. Wt 448
Purity >98%
Synonyms JTC801

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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