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- Lihao Gu, .et al. 10-Hydroxy-2-Decenoic Acid in Royal Jelly Extract Induced Both Filaggrin and Amino Acid in a Cultured Human Three-Dimensional Epidermis Model, Cosmetics, 2017, 4(4), 48
- Toshio Yawata, .et al. Brain opioid and nociceptin receptors are involved in regulation of bombesin-induced activation of central sympatho-adrenomedullary outflow in the rat, Mol Cell Biochem, 2016, Jan;411(1-2):201-11 PMID: 26427671
Biological Activity
JTC-801 is a selective antagonist for the nociceptin receptor, also known as the ORL-1 receptor.
| In vitro (25°C) | DMSO | 88 mg/mL (196.45 mM) | |
| Water | Insoluble | ||
| Ethanol | 30 mg/mL (66.97 mM) | ||
| In vivo | 0.5% methylcellulose | 28 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 22.32 mL | 111.61 mL | 223.21 mL |
| 0.5 mM | 4.46 mL | 22.32 mL | 44.64 mL |
| 1 mM | 2.23 mL | 11.16 mL | 22.32 mL |
| 5 mM | 0.45 mL | 2.23 mL | 4.46 mL |
*The above data is based on the productmolecular weight 448. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A11076 |
|---|---|
| Actions | Antagonist |
| CAS No. | 244218-51-7 |
| Formula | C26H25N3O2.HCl |
| M. Wt | 448 |
| Purity | >98% |
| Synonyms | JTC801 |
| SMILES | CCC1=CC=C(C=C1)OCC2=CC=CC=C2C(=O)NC3=CC4=C(C=C3)N=C(C=C4N)C.Cl |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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