Ketanserin (Vulketan Gel)

Catalog No.: A10497

5-HT2A serotonin receptor antagonist

Ketanserin (Vulketan Gel) Chemical Structure

CAS NO. 74050-98-9

Ketanserin (Vulketan Gel) is specific 5-HT2A serotonin receptor antagonist with a Ki of 2.5 nM for rat and human 5-HT2A.

Availability: In stock

Package Price Qty
50 mg
$40.00
100 mg
$60.00
250 mg
$120.00
500 mg
$220.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Ketanserin (Vulketan Gel) is specific 5-HT2A serotonin receptor antagonist with a Ki of 2.5 nM for rat and human 5-HT2A.
Targets
5-HT2A 5-HT2C (Rat) 5-HT2C (Human)
2.5 nM(Ki)50 nM(Ki)100 nM(Ki)
In vitro DMSO 2 mg/mL (5.05 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.29 mL 126.44 mL 252.89 mL
0.5 mM 5.06 mL 25.29 mL 50.58 mL
1 mM 2.53 mL 12.64 mL 25.29 mL
5 mM 0.51 mL 2.53 mL 5.06 mL

*The above data is based on the productmolecular weight 395.43. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A10497
Actions Antagonist
M. Wt 395.43
Formula C22H22FN3O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 74050-98-9
Synonyms R 41468, Vulketan Gel
SMILES C1CN(CCC1C(=O)C2=CC=C(C=C2)F)CCN3C(=O)C4=CC=CC=C4NC3=O

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