Keto-itraconazole

Name: Keto-itraconazole
Brand: Adooq Bioscience
SKU: A69803
Rating: 5 (288 reviews)

Catalog No.: A69803

CYP3A Inhibitor

Keto-itraconazole, a potent inhibitor of CYP3A, is a metabolite of Itraconazole. It demonstrates a significant unbound IC50 value of 4.6 nM when assessed using human liver microsomes in conjunction with midazolam. This compound is valuable for research focused on drug metabolism and interactions involving CYP3A-mediated pathways.

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Keto-itraconazole 112560-33-5 CYP3A Inhibitor

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Grouped product items
Size	Price	Stock
1mg	$250.00	In stock
2mg	$370.00	In stock
5mg	$880.00	In stock
10mg	$1,560.00	In stock
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Biological Activity

Description	Keto-itraconazole, a potent inhibitor of CYP3A, is a metabolite of Itraconazole. It demonstrates a significant unbound IC50 value of 4.6 nM when assessed using human liver microsomes in conjunction with midazolam. This compound is valuable for research focused on drug metabolism and interactions involving CYP3A-mediated pathways.

Product Information

Catalog Num	A69803
Formula	C35H36Cl2N8O5
Molecular Weight	719.62
CAS Number	112560-33-5
SMILES	O=C1N(N=CN1C2=CC=C(C=C2)N3CCN(CC3)C4=CC=C(C=C4)OC[C@@H]5O[C@](CN6N=CN=C6)(OC5)C7=CC=C(C=C7Cl)Cl)C(C)C(C)=O
Synonyms	keto-ITZ

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