Fig. 1 · Structure
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KSK94
H3 receptor Antagonist
KSK94 is a high-affinity antagonist of the histamine H3 receptor, exhibiting Ki values of 7.9 nM for H3, along with significant activity at sigma-1 and sigma-2 receptors at 2958 nM and 75.2 nM, respectively. This compound is utilized in research focused on nociceptive and neuropathic pain, providing insights into pain mechanisms and potential therapeutic interventions.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 2566716-07-0 |
| Applications | H3 receptor Antagonist |
| Formula | C25H26N4O |
| Molecular Weight | 398.50 |
| SMILES | N#CC(C=C1)=CC=C1C2=CC=C(OCCCN3CCN(C4=CC=NC=C4)CC3)C=C2 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.