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KSL 128114

Catalog No.: A84821
Syntenin Peptide Inhibitor
KSL 128114 is a potent peptide inhibitor of syntenin, targeting the PDZ1 domain with nanomolar affinity. This compound exhibits stability in human plasma and mouse hepatic microsomes, making it suitable for in vitro and in vivo studies. KSL 128114 demonstrates selective inhibition of syntenin, providing valuable insights into cellular signaling pathways and potential therapeutic applications in disorders associated with syntenin dysregulation.
KSL 128114 2757292-12-7 Syntenin Peptide Inhibitor
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Research use only. We do not sell to patients.
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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionKSL 128114 is a potent peptide inhibitor of syntenin, targeting the PDZ1 domain with nanomolar affinity. This compound exhibits stability in human plasma and mouse hepatic microsomes, making it suitable for in vitro and in vivo studies. KSL 128114 demonstrates selective inhibition of syntenin, providing valuable insights into cellular signaling pathways and potential therapeutic applications in disorders associated with syntenin dysregulation.
Product Information
Catalog NumA84821
FormulaC96H165N39O21
Molecular Weight2201.59
CAS Number2757292-12-7
SequenceAc-{d-Arg}-Arg-{d-Arg}-Gly-{d-Arg}-Lys-{d-Lys}-Arg-{d-Arg}-Ser-His-Trp-{Tle}-{Chg}-Asp-Ile
Sequence shorteningAc-{d-Arg}-R-{d-Arg}-G-{d-Arg}-K-{d-Lys}-R-{d-Arg}-SHW-{Tle}-{Chg}-DI
SMILESC([C@H](NC([C@H](CC1=CN=CN1)NC([C@@H](NC([C@H](NC([C@@H](NC([C@H](NC([C@@H](NC([C@H](NC(CNC([C@H](NC([C@@H](NC([C@@H](CCCNC(=N)N)NC(C)=O)=O)CCCNC(=N)N)=O)CCCNC(=N)N)=O)=O)CCCNC(=N)N)=O)CCCCN)=O)CCCCN)=O)CCCNC(=N)N)=O)CCCNC(=N)N)=O)CO)=O)=O)C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@@H]([C@H](CC)C)C(O)=O)=O)CC(O)=O)=O)C2CCCCC2)=O)[C@](C)(C)C)=O)C=3C=4C(NC3)=CC=CC4
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