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LDLRAP1-IN-1

LDLRAP1 Inhibitor

LDLRAP1-IN-1 is an inhibitor of LDLRAP1, targeting the interaction between LDLRAP1 and LDL receptor (LDLR) with an IC50 of 4.98 μM. This compound covalently modifies the C119 residue at the LDLRAP1-LDLR binding interface, effectively disrupting their interaction. Additionally, LDLRAP1-IN-1 demonstrates antiviral activity against HCoV-OC43, making it a valuable tool for research in lipid metabolism and antiviral studies.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Inhibitor
CAS Number	3093624-24-6
Applications	LDLRAP1 Inhibitor
Formula	C₂₁H₁₄ClN₅O₄
Molecular Weight	435.82
SMILES	O=C(NC1=CC=C(N2N=CN=C2)C=C1)C3=CC([N+]([O-])=O)=CC=C3OC4=CC=C(Cl)C=C4

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.