lumateperone Tosylate

Catalog No.: A12279

5-HT2A receptor antagonist

lumateperone Tosylate

lumateperone Tosylate Chemical Structure

CAS NO. 1187020-80-9

Lumateperone Tosylate is a 5-HT2A receptor antagonist (Ki = 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki = 32 nM), and a SERT blocker (Ki = 61 nM).

Availability: In stock

Package Price Qty
5 mg
$108.00
10 mg
$186.00
50 mg
$552.00
100 mg
$1,104.00
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Biological Activity

Lumateperone Tosylate is a 5-HT2A receptor antagonist (Ki = 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki = 32 nM), and a SERT blocker (Ki = 61 nM).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.68 mL 88.39 mL 176.77 mL
0.5 mM 3.54 mL 17.68 mL 35.35 mL
1 mM 1.77 mL 8.84 mL 17.68 mL
5 mM 0.35 mL 1.77 mL 3.54 mL

*The above data is based on the productmolecular weight 565.7. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12279
Actions Antagonist
CAS No. 1187020-80-9
Formula C31H36FN3O4S
M. Wt 565.7
Purity >98%
Synonyms ITI-007, ITI007, ITI 007
SMILES O=C(C1=CC=C(F)C=C1)CCCN2CC[[email protected]@](N3CCN(C)C4=C3C5=CC=C4)([H])[[email protected]@]5([H])C2.O=S(C6=CC=C(C)C=C6)(O)=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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