Fig. 1 · Structure
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Lupanine perchlorate
nAChR Inhibitor
Lupanine perchlorate is a natural ketonic derivative of sparteine that functions as an nAChR inhibitor. It exhibits significant ganglioplegic activity and demonstrates a binding affinity for nicotinic receptors with a Ki value of 500 nM. This compound is commonly utilized in research focused on studying neuronal signaling and the effects of cholinergic modulation.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 7400-11-5 |
| Applications | nAChR Inhibitor |
| Formula | C15H25ClN2O5 |
| Molecular Weight | 348.82 |
| Synonyms | D-Lupanine perchlorate |
| SMILES | O=C1N2[C@]([C@](C3)([H])CN(CCCC4)[C@]4([H])[C@]3([H])C2)([H])CCC1.O=Cl(=O)(O)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.