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LY215840

Catalog No.: A29779
5-HT2/5-HT7 Antagonist
LY215840 is a selective antagonist of the 5-HT2 and 5-HT7 serotonin receptors. This compound effectively inhibits serotonin-induced vasorelaxation in the canine coronary artery, demonstrating significant potential for research in cardiovascular pharmacology and serotonin receptor signaling. Its application extends to studies exploring the role of serotonin receptors in various physiological and pathological processes.
LY215840 137328-52-0 5-HT2/5-HT7 Antagonist
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Research use only. We do not sell to patients.
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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionLY215840 is a selective antagonist of the 5-HT2 and 5-HT7 serotonin receptors. This compound effectively inhibits serotonin-induced vasorelaxation in the canine coronary artery, demonstrating significant potential for research in cardiovascular pharmacology and serotonin receptor signaling. Its application extends to studies exploring the role of serotonin receptors in various physiological and pathological processes.
Product Information
Catalog NumA29779
FormulaC24H33N3O2
Molecular Weight395.54
CAS Number137328-52-0
SMILESCC(N1C2=CC=CC3=C2C(C[C@]4([H])[C@]3([H])C[C@@H](C(N[C@@H]5[C@@H](CCC5)O)=O)CN4C)=C1)C
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GPCR/G Protein > 5-HT Receptors